Pharmaceutical Raw Materials Tasimelteon Hetlioz For Good Sleep
Tasimelteon Basic Info
Tasimelteon Name Tasimelteon
Tasimelteon Purity: >99%
Tasimelteon CAS: 609799-22-6
Tasimelteon Molecular Weight: 245.322
Tasimelteon Certification: ISO 9001, USP, BP
Tasimelteon State: Solid
Tasimelteon Appearance: White Crystalline Powder
Tasimelteon Mf: C15h19no2
Tasimelteon Boiling Point: 442.553°c
What is Tasimelteon?
Tasimelteon is a melatonin receptor agonist. It works by targeting receptors in the brain that control the timing of the sleep-wake cycle. In clinical trials, totally blind individuals with Non-24 who were treated with tasimelteon slept longer during the night. Tasimelteon was also found to decrease the amount of time totally blind individuals with Non-24 slept during the day.
Tasimelteon vs Ramelteon
Uses. Both drug treat sleep disorders. Tasimelteon is approved for Non-24-Hour Sleep-Wake Disorder, ramelteon is approved for insomnia (difficulty falling asleep).
Mechanism. Both bind melatonin receptors
Receptor binding. Tasimelteon has 2-5x greater affinity for the melatonin receptor MT2 than MT1. Ramelteon has 10x the affinity for the melatonin receptor MT1 than MT2.
Half-life. The half-life of tasimelteon is about 1 hour (according to one source). The half-life of ramelteon is 1-2.6 hours.
Interactions. Ramelteon has drug-drug interactions with Amiodarone, Ciprofloxacin, Fluvoxamine, Ticlopidine. Since tasimelteon is metabolized by CYP1A2 and CYP3A4/5, it interactions with many drug also metabolized by these enzymes.
The dose of this medicine will be different for different patients. Follow your doctor's orders or the directions on the label. The following information includes only the average doses of this medicine. If your dose is different, do not change it unless your doctor tells you to do so.
The amount of medicine that you take depends on the strength of the medicine. Also, the number of doses you take each day, the time allowed between doses, and the length of time you take the medicine depend on the medical problem for which you are using the medicine.
For oral dosage form (capsules):
For non-24-hour sleep-wake disorder:
Adults—20 milligrams (mg) per day, taken before bedtime.
Children—Use and dose must be determined by your doctor.
|Appearance||White to off-white crystalline powder||Complies|
|Loss on drying||≤0.5%||0.01%|
|Residue on Ignition||≤0.1%||0.01%|
|Related Substances (HPLC)||Impurity A≤0.1%|
Any other single impurity≤0.1%
|Chiral Purity (HPLC)||≥99.9%||100%|
|Assay||98.0 - 102.0% ( on anhydrous basis)||100.2%|
|Conclusion||Complies with the Enterprise Standard.|
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